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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- B2176 GSK1059615Target: PI3K|mTORSummary: PI3K和mTOR抑制剂
- A8354 A66Target: PI3KSummary: P110α抑制剂
- A4097 CUDC-907中文名: 非美诺司他Target: Histone Deacetylases (HDACs)|PI3KSummary: PI3K/HDAC抑制剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- A8556 GSK21264581 CitationTarget: PI3K|mTORSummary: PI3K/mTOR抑制剂
- B1036 MLN49245 CitationTarget: NAE|Ubiquitin-activating Enzyme E1|SUMOylationSummary: NAE抑制剂
- B4894 SP2509Target: Histone DemethylasesSummary: 新型LSD1拮抗剂
- B1579 JIB-041 CitationTarget: Histone DemethylasesSummary: Jumonji组蛋白去甲基化酶抑制剂