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- B1250 Ezatiostat hydrochloride3 CitationTarget: Gutathione S-transferaseSummary: GST抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A8225 EzatiostatTarget: Gutathione S-transferaseSummary: (GST) P1-1抑制剂
- A1947 MEK162 (ARRY-162, ARRY-438162)中文名: 贝美替尼Target: MEKSummary: MEK1/2抑制剂
- A3887 Trametinib DMSO solvate1 CitationTarget: MEKSummary: 变构MEK1/MEK2 激酶抑制剂
- A1337 U0126-EtOH10 CitationTarget: MEKSummary: MEK1/2抑制剂
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂
- A3018 Trametinib (GSK1120212)7 Citation中文名: 曲美替尼Target: MEKSummary: MEK1和MEK2抑制剂
- A5707 PD318088Target: MEKSummary: MEK1/2变构抑制剂
- A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2抑制剂