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- A8716 LY3009120Target: RafSummary: Pan-RAF和RAF二聚体抑制剂
- B6801 SCH 79797 dihydrochlorideTarget: PARsSummary: PAR1受体拮抗剂
- B1174 LGX818中文名: 康奈非尼Target: RafSummary: RAF抑制剂
- A4228 Nutlin-3Target: MDM2Summary: MDM2 拮抗剂
- A3347 Dabrafenib Mesylate (GSK-2118436)中文名: 达帕菲尼甲磺酸盐Target: RafSummary: BRAF(V600E)抑制剂
- A3762 RG71125 CitationTarget: MDM2Summary: MDM2抑制剂
- N1315 Parthenolide中文名: 小白菊内酯,欧苷菊Target: Histone Deacetylases (HDACs)|MDM2|DNA Methyltransferases|p53|5-HT
- A5071 GDC-08791 CitationTarget: RafSummary: B-Raf抑制剂
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- A3009 Sorafenib2 Citation中文名: 索拉非尼Target: Raf|VEGFRSummary: Raf激酶和酪氨酸激酶抑制剂