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- A8626 ETP-46464Target: PI3K|mTOR|DNA-PK|ATM/ATRSummary: ATR抑制剂
- A2574 Aprotinin1 Citation中文名: 抑酶肽Target: Trypsin|Chymotrypsin|Kallikrein|TrypsinogenSummary: 牛胰蛋白酶抑制剂
- B1135 GDC-0623Target: MEKSummary: MEK1抑制剂
- A8312 Torin 17 CitationTarget: mTORSummary: MTOR抑制剂
- A5078 KU-0063794Target: mTORSummary: mTORC1和mTORC2的抑制剂
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂
- B2172 PP121Target: mTOR|Eph Receptors|VEGFR|PDGFR|Bcr-Abl|Src|DNA-PK|P110|HckSummary: 酪氨酸激酶和磷酸肌醇激酶双重抑制剂
- A8488 NVP-BGT226Target: PI3K|mTORSummary: 新型的PI3K/mTOR选择性抑制剂
- A1947 MEK162 (ARRY-162, ARRY-438162)中文名: 贝美替尼Target: MEKSummary: MEK1/2抑制剂
- B1267 RefametinibTarget: MEKSummary: MEK1/MEK2抑制剂