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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A3248 BMS345541 hydrochlorideTarget: IKKSummary: IKK抑制剂
- B1387 (-)-Blebbistatin3 Citation中文名: 布雷他汀Target: Myosin II ATPasesSummary: 非肌肉肌球蛋白II型ATP酶抑制剂
- A5161 Imiquimod中文名: 咪喹莫特Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂,具有抗病毒和抗肿瘤活性的免疫调节剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- B5996 Motolimod (VTX-2337)Target: Toll-like receptors (TLRs)Summary: TLR8激动剂
- B5551 Poly(I:C)Target: Toll-like receptors (TLRs)Summary: Toll样受体3(TLR3)激动剂
- A3444 GS-9620中文名: 维沙莫德Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂
- B1054 Resiquimod (R-848)2 Citation中文名: 雷西莫特,瑞喹莫德Target: Toll-like receptors (TLRs)Summary: 免疫应答调节剂