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- B5854 Pexidartinib (PLX3397)3 Citation中文名: 培西达替尼Target: FLT3|c-Kit|CSF1RSummary: CSF-1R抑制剂
- A8715 SBI-02069652 CitationTarget: ULK1Summary: ULK1抑制剂
- B6962 CMPD-1Target: Microtubules/Tubulins|MK2Summary: p38α介导的MK2a磷酸化的抑制剂
- A8335 Palbociclib (PD0332991) Isethionate1 Citation中文名: 帕博西尼羟乙基磺酸盐Target: Cyclin-Dependent KinasesSummary: CDK4/6抑制剂
- A4512 Cucurbitacin I中文名: 葫芦素 ITarget: STAT|JAKSummary: STAT3/JAK2信号转导抑制剂
- A4224 GDC-01522 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: IAP 拮抗剂
- A8210 GDC-094110 CitationTarget: PI3KSummary: PI3K抑制剂
- A8217 ICG 0011 CitationSummary: Wnt/β-catenin信号通路的抑制剂
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂