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- N2791 Cucurbitacin E中文名: 葫芦素 ETarget: ActinSummary: 抑制肌动蛋白解聚
- B1642 WYE-125132 (WYE-132)Target: mTORSummary: mTOR抑制剂
- A1987 Ki164254 CitationTarget: LPA ReceptorsSummary: LPA受体拮抗剂
- B4492 HS-173Target: PI3KSummary: PI3Kα抑制剂
- B2307 LGK-9741 CitationSummary: PORCN抑制剂
- A2678 SU112742 CitationTarget: METSummary: C-Met抑制剂
- B1286 AZD7545Target: PDHKSummary: 有效的PDHK选择性抑制剂
- A4180 SRT1720 HCl3 CitationTarget: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT1激活剂
- A8245 Sorafenib Tosylate1 Citation中文名: 甲苯磺酸索拉非尼Target: Raf|VEGFRSummary: Raf激酶和酪氨酸激酶抑制剂
- A8173 Romidepsin (FK228, depsipeptide)7 Citation中文名: 罗米地辛Target: Histone Deacetylases (HDACs)Summary: 选择性的HDAC1/HDAC2抑制剂