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Signaling Pathways - Voltage-gated Sodium (NaV) Channels - FLT3

29件产品中的 1-10

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  1. Dovitinib (TKI258) Lactate
    B5953 Dovitinib (TKI258) Lactate
    Target: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFR
    Summary: 酪氨酸激酶抑制剂(TKI)
      ≥10.62 mg/mL
      ≥168.2 mg/mL
  2. Pexidartinib (PLX3397)
    B5854 Pexidartinib (PLX3397)
     3 Citation
    中文名: 培西达替尼
    Target: FLT3|c-Kit|CSF1R
    Summary: CSF-1R抑制剂
      ≥20.9 mg/mL
      insoluble in H2O
  3. AZD2932
    B5835 AZD2932
    Target: FLT3|VEGFR|PDGFR|c-Kit
    Summary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
      Soluble in DMSO
  4. Altiratinib
    B5832 Altiratinib
     1 Citation
    Target: FLT3|VEGFR|Trk Receptors|c-MET|Tie-2
    Summary: c-MET/TIE-2/VEGFR抑制剂
      ≥21.55 mg/mL
      insoluble in H2O
  5. UNC2025
    B8016 UNC2025
     1 Citation
    Target: MER|FLT3
    Summary: 口服生物可利用的双重MER/FLT3抑制剂
      ≥23.85 mg/mL
      ≥6.09 mg/mL
  6. G-749
    A8889 G-749
    Target: Aurora Kinases|FLT3|c-RET
    Summary: FLT3抑制剂
      ≥26.05 mg/mL
      insoluble in H2O
  7. ProTx II
    B5515 ProTx II
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: NaV1.7通道阻断剂
      Soluble to 1 mg/mL
  8. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  9. Amiloride HCl dihydrate
    B2268 Amiloride HCl dihydrate
    中文名: 盐酸阿米洛利二水合物
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Urokinases
    Summary: 有效上皮钠通道(ENaC)阻断剂
      ≥14.05 mg/mL
      insoluble in H2O
  10. Bupivacaine HCl
    B1420 Bupivacaine HCl
    中文名: 盐酸布比卡因
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 麻醉药
      ≥10.25 mg/mL
      ≥16.23 mg/mL

29件产品中的 1-10

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