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Signaling Pathways - DCLK2 - Nrf2/ARE signal - Aromatases - P-glycoprotein (P-gp)

10 件产品

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  1. Anastrozole
    B1382 Anastrozole
    中文名: 阿那曲唑
    Target: Aromatases
    Summary: 芳香酶抑制剂
      ≥14.15 mg/mL
      insoluble in H2O
  2. LY335979 (Zosuquidar 3HCL)
    A8549 LY335979 (Zosuquidar 3HCL)
     1 Citation
    中文名: 唑喹达三盐酸盐
    Target: P-glycoprotein (P-gp)
    Summary: Pgb(P糖蛋白)抑制剂
      ≥17.1 mg/mL
      ≥31.9 mg/mL
  3. Letrozole
    A1307 Letrozole
    中文名: 来曲唑
    Target: Aromatases
    Summary: 非甾体类芳香酶抑制剂。
      ≥14.265 mg/mL
      insoluble in H2O
  4. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  5. Tariquidar methanesulfonate, hydrate
    A3859 Tariquidar methanesulfonate, hydrate
    中文名: 他立喹达二甲磺酸盐六水合物
    Target: P-glycoprotein (P-gp)
    Summary: P-糖蛋白抑制剂
      ≥56.2 mg/mL
      insoluble in H2O
  6. LRRK2-IN-1
    A3558 LRRK2-IN-1
     1 Citation
    Target: LRRK2|DCLK2
    Summary: LRRK2抑制剂
      ≥28.55 mg/mL
      insoluble in H2O
  7. Elacridar
    A3384 Elacridar
    中文名: 依克立达
    Target: P-glycoprotein (P-gp)
    Summary: BCRP抑制剂
      ≥56.4 mg/mL
      insoluble in H2O
  8. Tariquidar
    A8208 Tariquidar
     2 Citation
    中文名: 他立喹达
    Target: P-glycoprotein (P-gp)
    Summary: P-糖蛋白抑制剂
      ≥16.17 mg/mL
      insoluble in H2O
  9. GDC-0449 (Vismodegib)
    A3021 GDC-0449 (Vismodegib)
     1 Citation
    中文名: 维莫德吉
    Target: P-glycoprotein (P-gp)|Hedgehog
    Summary: Hedgehog拮抗剂
      ≥21.08 mg/mL
      insoluble in H2O
  10. 5,7-dihydroxychromone
    N2172 5,7-dihydroxychromone
     1 Citation
    中文名: 5,7-二羟基色酮
    Target: Nrf2/ARE signal|PPAR
    Summary: Nrf2/ARE信号激活剂和PPARγ激动剂
      ≥7.05 mg/mL
      insoluble in H2O

10 件产品

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