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Signaling Pathways - Pregnane X receptor(PXR) - JAK - PDHK - Calcium-Activated Potassium (KCa) Channels

27件产品中的 1-10

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  1. Cerdulatinib (PRT062070)
    B8023 Cerdulatinib (PRT062070)
    Target: JAK|Syk|TYK2
    Summary: Syk/JAK抑制剂
      ≥22.3 mg/mL
      insoluble in H2O
  2. Dequalinium Chloride
    B2191 Dequalinium Chloride
    中文名: 地喹氯铵
    Target: PKC|Calcium-Activated Potassium (KCa) Channels
    Summary: PKC抑制剂
      insoluble in DMSO
      insoluble in H2O
  3. GLPG0634
    B1130 GLPG0634
     1 Citation
    中文名: 菲戈替尼
    Target: JAK
    Summary: JAK1抑制剂
      ≥21.3 mg/mL
      insoluble in H2O
  4. AZD7545
    B1286 AZD7545
    Target: PDHK
    Summary: 有效的PDHK选择性抑制剂
      ≥21.85 mg/mL
      insoluble in H2O
  5. Lithocholic Acid
    A8463 Lithocholic Acid
    中文名: 石胆酸
    Target: Farnesoid X receptors (FXRs)|Vitamin D receptors (VDRs)|Pregnane X receptor(PXR)
    Summary: 维生素D受体PXR和FXR的激活剂
      ≥12.95 mg/mL
      insoluble in H2O
  6. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  7. TRAM-34
    A1888 TRAM-34
    Target: Calcium-Activated Potassium (KCa) Channels
    Summary: KCa3.1阻断剂
      ≥17.25 mg/mL
      insoluble in H2O
  8. PP 1
    A8215 PP 1
    Target: Src|EGFR|JAK|ZAP-70
    Summary: Src家族酪氨酸激酶抑制剂
      ≥7.03 mg/mL
      insoluble in H2O
  9. Cucurbitacin I
    A4512 Cucurbitacin I
    中文名: 葫芦素 I
    Target: STAT|JAK
    Summary: STAT3/JAK2信号转导抑制剂
      ≥22.45 mg/mL
      ≥51.2 mg/mL
  10. Cercosporamide
    A4511 Cercosporamide
    中文名: 尾孢素酰胺
    Target: JAK|MNK
    Summary: Mnk2和JAK3抑制剂
      soluble in DMSO

27件产品中的 1-10

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