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Signaling Pathways - NPFF receptor - Bromodomain and Extra-Terminal motif (BET) - M3 Receptors - P-glycoprotein (P-gp)

12件产品中的 1-10

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  1. BIBP 3226 trifluoroacetate
    B7155 BIBP 3226 trifluoroacetate
    Target: NPY Receptors|NPFF receptor
    Summary: 混合NPY Y1和NPFF受体拮抗剂
      ≥78 mg/mL
      ≥12.13 mg/mL
  2. Otilonium Bromide
    B1607 Otilonium Bromide
    中文名: 奥替溴铵
    Target: M3 Receptors
    Summary: AChR抑制剂
      ≥28.18 mg/mL
      ≥55.8 mg/mL
  3. Darifenacin HBr
    B1600 Darifenacin HBr
    中文名: 氢溴酸达非那新
    Target: M3 Receptors
    Summary: 选择性M3毒蕈碱受体拮抗剂
      ≥20.2 mg/mL
      insoluble in H2O
  4. Solifenacin succinate
    B1614 Solifenacin succinate
    中文名: 琥珀酸索非那新
    Target: M3 Receptors
    Summary: 毒蕈碱受体拮抗剂
      ≥24.05 mg/mL
      ≥53.6 mg/mL
  5. I-BET151 (GSK1210151A)
    B1500 I-BET151 (GSK1210151A)
     2 Citation
    Target: Bromodomain and Extra-Terminal motif (BET)
    Summary: BET的选择性抑制剂
      ≥41.5 mg/mL
      insoluble in H2O
  6. LY335979 (Zosuquidar 3HCL)
    A8549 LY335979 (Zosuquidar 3HCL)
     1 Citation
    中文名: 唑喹达三盐酸盐
    Target: P-glycoprotein (P-gp)
    Summary: Pgb(P糖蛋白)抑制剂
      ≥17.1 mg/mL
      ≥31.9 mg/mL
  7. Atropine sulfate monohydrate
    A8369 Atropine sulfate monohydrate
    中文名: 硫酸阿托品一水合物
    Target: M3 Receptors|M1 Receptors|M2 Receptors|M4 Receptors|M5 Receptors
    Summary: MAChRs拮抗剂
      ≥34.74 mg/mL
      ≥56.5 mg/mL
  8. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  9. Tariquidar methanesulfonate, hydrate
    A3859 Tariquidar methanesulfonate, hydrate
    中文名: 他立喹达二甲磺酸盐六水合物
    Target: P-glycoprotein (P-gp)
    Summary: P-糖蛋白抑制剂
      ≥56.2 mg/mL
      insoluble in H2O
  10. Elacridar
    A3384 Elacridar
    中文名: 依克立达
    Target: P-glycoprotein (P-gp)
    Summary: BCRP抑制剂
      ≥56.4 mg/mL
      insoluble in H2O

12件产品中的 1-10

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