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Signaling Pathways - Aldehyde Dehydrogenases - 5-HT2 Receptor - P-glycoprotein (P-gp) - Cytochrome P450 (CYP450)

23件产品中的 1-10

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  1. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  2. Alda 1
    B5508 Alda 1
    Target: Aldehyde Dehydrogenases
    Summary: ALDH2激活剂
      ≥15.15 mg/mL
      insoluble in H2O
  3. SCH 23390 hydrochloride
    B6506 SCH 23390 hydrochloride
    Target: dopamine receptor|5-HT1 Receptor|5-HT2 Receptor
    Summary: 多巴胺受体拮抗剂
      Soluble to 100 mM in sterile water and to 50 mM in ethanol
  4. Methylergometrine maleate
    B6347 Methylergometrine maleate
    中文名: 马来酸甲麦角新碱
    Target: 5-HT1 Receptor|5-HT2 Receptor
    Summary: 5-HT1/5-HT2受体拮抗剂
      Soluble to 25 mM in H2O
  5. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  6. Fluconazole
    B2094 Fluconazole
    中文名: 氟康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 三唑抗真菌剂
      ≥10.9 mg/mL
      insoluble in H2O
  7. Rifabutin
    B2126 Rifabutin
    中文名: 利福布丁
    Target: Cytochrome P450 (CYP450)
    Summary: 抗结核药物
      ≥42.35 mg/mL
      insoluble in H2O
  8. TOK-001
    A8623 TOK-001
    中文名: 加来特龙,伽来特隆
    Target: Androgen Receptors|Cytochrome P450 (CYP450)
    Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
      ≥12.4 mg/mL
      insoluble in H2O
  9. LY335979 (Zosuquidar 3HCL)
    A8549 LY335979 (Zosuquidar 3HCL)
     1 Citation
    中文名: 唑喹达三盐酸盐
    Target: P-glycoprotein (P-gp)
    Summary: Pgb(P糖蛋白)抑制剂
      ≥17.1 mg/mL
      ≥31.9 mg/mL
  10. Clotrimazole
    A8401 Clotrimazole
     2 Citation
    中文名: 克霉唑
    Target: Cytochrome P450 (CYP450)
    Summary: 抗真菌化合物
      ≥28.1 mg/mL
      insoluble in H2O

23件产品中的 1-10

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