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Signaling Pathways - MDM2 - NADPH Oxidases - Trk Receptors - Cytochrome P450 (CYP450)

27件产品中的 1-10

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  1. GKT137831
    B4763 GKT137831
     1 Citation
    Target: NADPH Oxidases
    Summary: Nox1/Nox4双重抑制剂
      ≥39.5 mg/mL
      insoluble in H2O
  2. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  3. Entrectinib
    B5859 Entrectinib
    中文名: 恩曲替尼
    Target: Trk Receptors|ALK|ROS1
    Summary: ALK激酶抑制剂
      ≥28.05 mg/mL
      insoluble in H2O
  4. Altiratinib
    B5832 Altiratinib
     1 Citation
    Target: FLT3|VEGFR|Trk Receptors|c-MET|Tie-2
    Summary: c-MET/TIE-2/VEGFR抑制剂
      ≥21.55 mg/mL
      insoluble in H2O
  5. ANA 12
    B5712 ANA 12
     1 Citation
    Target: Trk Receptors
    Summary: TrkB受体拮抗剂
      ≥10.175 mg/mL
      insoluble in H2O
  6. Diphenyleneiodonium chloride
    B6326 Diphenyleneiodonium chloride
    中文名: 二苯基氯化碘盐
    Target: NADPH Oxidases|NOS|GPR3
    Summary: iNOS和eNOS抑制剂,GPR3激动剂
      ≥6.99 mg/mL
      insoluble in H2O
  7. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  8. Apocynin
    B3675 Apocynin
    中文名: 罗布麻宁,夹竹桃麻素,香兰基甲基酮
    Target: NADPH Oxidases
    Summary: 选择性NADPH氧化酶抑制剂
      ≥8.25 mg/mL
  9. Amitriptyline HCl
    B2231 Amitriptyline HCl
    中文名: 盐酸阿米替林
    Target: Trk Receptors|5-HT2 Receptors|Norepinephrine transporter|5-HT Transporters
    Summary: 血清素/去甲肾上腺素受体/5-HT4/5-HT2抑制剂
      ≥15.69 mg/mL
      ≥43.9 mg/mL
  10. Fluconazole
    B2094 Fluconazole
    中文名: 氟康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 三唑抗真菌剂
      ≥10.9 mg/mL
      insoluble in H2O

27件产品中的 1-10

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