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Signaling Pathways - Insulin and Insulin-like Receptors - CysLT1 - CREBBP - Vitamin D receptors (VDRs)

13件产品中的 1-10

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  1. MK-571 sodium salt hydrate
    B8031 MK-571 sodium salt hydrate
     3 Citation
    Target: CysLT1
    Summary: CysLT1受体拮抗剂
      ≥10.3 mg/mL
      ≥122.2 mg/mL
  2. Calcifediol
    B2140 Calcifediol
    中文名: 骨化二醇
    Target: Vitamin D receptors (VDRs)
    Summary: 维生素D3的主要循环形式
      ≥13.65 mg/mL
      insoluble in H2O
  3. Doxercalciferol
    B2091 Doxercalciferol
     1 Citation
    中文名: 度骨化醇
    Target: Vitamin D receptors (VDRs)
    Summary: 维生素D受体激活剂
      ≥11.5 mg/mL
      insoluble in H2O
  4. Lithocholic Acid
    A8463 Lithocholic Acid
    中文名: 石胆酸
    Target: Farnesoid X receptors (FXRs)|Vitamin D receptors (VDRs)|Pregnane X receptor(PXR)
    Summary: 维生素D受体PXR和FXR的激活剂
      ≥12.95 mg/mL
      insoluble in H2O
  5. GSK1838705A
    A8440 GSK1838705A
    Target: Insulin and Insulin-like Receptors|ALK
    Summary: ATP竞争性IGF-IR/IR/ALK抑制剂
      ≥26.65 mg/mL
      insoluble in H2O
  6. GSK1904529A
    A1302 GSK1904529A
    Target: Insulin and Insulin-like Receptors
    Summary: IGF-1R/IR 选择性抑制剂
      ≥42.6 mg/mL
      insoluble in H2O
  7. BMS-754807
    A1185 BMS-754807
    Target: Insulin and Insulin-like Receptors
    Summary: 有效的、选择性的IGF-1R和InsR抑制剂
      ≥23.05 mg/mL
      insoluble in H2O
  8. SGC-CBP30
    A4491 SGC-CBP30
     2 Citation
    Target: CREBBP|EP300
    Summary: CREBBP/EP300 bromodomain抑制剂
      ≥20.05 mg/mL
      ≥4.67 mg/mL
  9. I-CBP 112
    A4490 I-CBP 112
    Target: CREBBP|EP300
    Summary: CBP/EP300 bromodomain抑制剂
      ≥49.6 mg/mL
      insoluble in H2O
  10. MK 0893
    A3608 MK 0893
    Target: Insulin and Insulin-like Receptors|Glucagon Receptors
    Summary: 胰高血糖素受体/ IGF-1R拮抗剂
      ≥24.05 mg/mL
      insoluble in H2O

13件产品中的 1-10

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