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Signaling Pathways - Cytochrome P450 (CYP450) - sodium channels - ALK - Ca2 /calmodulin-dependent protein kinases (CaMKs)

32件产品中的 1-10

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  1. β-Pompilidotoxin
    A1132 β-Pompilidotoxin
    Target: sodium channels
    Summary: 减慢Na+通道失活。
      ≥155.8 mg/mL
      ≥22.05 mg/mL
  2. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  3. Entrectinib
    B5859 Entrectinib
    中文名: 恩曲替尼
    Target: Trk Receptors|ALK|ROS1
    Summary: ALK激酶抑制剂
      ≥28.05 mg/mL
      insoluble in H2O
  4. KN-93 Phosphate
    B4969 KN-93 Phosphate
    Target: Ca2 /calmodulin-dependent protein kinases (CaMKs)
    Summary: CaM激酶II抑制剂
      ≥29.95 mg/mL
      ≥20.7 mg/mL
  5. PF-06463922
    B4882 PF-06463922
    中文名: 劳拉替尼
    Target: ALK|ROS1
    Summary: ALK/ROS1的强效选择性抑制剂
      ≥20.3 mg/mL
      insoluble in H2O
  6. Rottlerin
    B6803 Rottlerin
     1 Citation
    中文名: 揪毒素
    Target: PKC|Ca2 /calmodulin-dependent protein kinases (CaMKs)|PRAK|MAPKAP-K2
    Summary: PKC抑制剂
      ≥23.6 mg/mL
      insoluble in H2O
  7. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  8. Autocamtide-2-related inhibitory peptide
    B6831 Autocamtide-2-related inhibitory peptide
    Target: Ca2 /calmodulin-dependent protein kinases (CaMKs)
    Summary: 钙调蛋白依赖性蛋白激酶II(CaM激酶II,CaMKII)抑制剂
      ≥40.2 mg/mL
      ≥45.7 mg/mL
  9. Fluconazole
    B2094 Fluconazole
    中文名: 氟康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 三唑抗真菌剂
      ≥10.9 mg/mL
      insoluble in H2O
  10. Rifabutin
    B2126 Rifabutin
    中文名: 利福布丁
    Target: Cytochrome P450 (CYP450)
    Summary: 抗结核药物
      ≥42.35 mg/mL
      insoluble in H2O

32件产品中的 1-10

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