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Signaling Pathways - Cytochrome P450 (CYP450) - sodium channels - ALK - Estrogen and Related Receptors

35件产品中的 1-10

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  1. β-Pompilidotoxin
    A1132 β-Pompilidotoxin
    Target: sodium channels
    Summary: 减慢Na+通道失活。
      ≥155.8 mg/mL
      ≥22.05 mg/mL
  2. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  3. Entrectinib
    B5859 Entrectinib
    中文名: 恩曲替尼
    Target: Trk Receptors|ALK|ROS1
    Summary: ALK激酶抑制剂
      ≥28.05 mg/mL
      insoluble in H2O
  4. PF-06463922
    B4882 PF-06463922
    中文名: 劳拉替尼
    Target: ALK|ROS1
    Summary: ALK/ROS1的强效选择性抑制剂
      ≥20.3 mg/mL
      insoluble in H2O
  5. (Z)-4-Hydroxytamoxifen
    B5421 (Z)-4-Hydroxytamoxifen
    中文名: 4-羟基他莫昔芬
    Target: Estrogen and Related Receptors
    Summary: 雌激素受体(ER)调节剂
      ≥38.8 mg/mL
      insoluble in H2O
  6. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  7. Erteberel (LY500307)
    B1518 Erteberel (LY500307)
    Target: Estrogen and Related Receptors
    Summary: ERβ激动剂
      ≥14.1 mg/mL
      insoluble in H2O
  8. Estriol
    B1507 Estriol
    中文名: 雌三醇
    Target: Estrogen and Related Receptors
    Summary: 雌激素受体拮抗剂
      ≥9.25 mg/mL
      insoluble in H2O
  9. Estradiol valerate
    B1506 Estradiol valerate
    中文名: 戊酸雌二醇
    Target: Estrogen and Related Receptors
    Summary: 雌激素受体激动剂
      ≥15.45 mg/mL
      insoluble in H2O
  10. Bazedoxifene HCl
    B1519 Bazedoxifene HCl
    中文名: 盐酸巴多昔芬
    Target: Estrogen and Related Receptors
    Summary: 新的非甾体,基于吲哚的雌激素受体调节剂(SERM)
      ≥25.35 mg/mL

35件产品中的 1-10

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