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- B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
- A8550 Telatinib (BAY 57-9352)中文名: 替拉替尼Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3、PDGFR-β和c-Kit抑制剂
- B1614 Solifenacin succinate中文名: 琥珀酸索非那新Target: M3 ReceptorsSummary: 毒蕈碱受体拮抗剂
- A4351 PluriSIn #1 (NSC 14613)Target: Stearoyl-CoA 9-desaturase (SCD-1)Summary: SCD1抑制剂
- A2168 Dovitinib (TKI-258, CHIR-258)2 Citation中文名: 多韦替尼Target: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: 多靶点RTK抑制剂
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- A8370 Axitinib (AG 013736)1 Citation中文名: 阿西替尼Target: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit抑制剂
- B1600 Darifenacin HBr中文名: 氢溴酸达非那新Target: M3 ReceptorsSummary: 选择性M3毒蕈碱受体拮抗剂
- B3607 A9395721 CitationTarget: Stearoyl-CoA 9-desaturase (SCD-1)Summary: 硬脂酰辅酶A去饱和酶1(SCD1)抑制剂
- B1607 Otilonium Bromide中文名: 奥替溴铵Target: M3 ReceptorsSummary: AChR抑制剂