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- A3742 Pyridostatin2 CitationTarget: G-quadruplexesSummary: 促生长停滞药物
- B6803 Rottlerin1 Citation中文名: 揪毒素Target: PKC|Ca2 /calmodulin-dependent protein kinases (CaMKs)|PRAK|MAPKAP-K2Summary: PKC抑制剂
- B5946 EW-71971 CitationTarget: BMP and Other Activin ReceptorsSummary: TGF-β I型受体激酶抑制剂
- A3392 Emodin中文名: 大黄素Target: CK2Summary: 天然存在的蒽醌,抗增殖
- B2114 Mitoxantrone HCl中文名: 米托蒽醌Target: Pim|Topoisomerases|USP|HIV IntegrasesSummary: 拓扑异构酶II抑制剂
- B2169 IPA-31 CitationTarget: PAKSummary: 非竞争性Pak1抑制剂
- A1794 LY2835219中文名: 甲磺酸阿贝西尼Target: Cyclin-Dependent KinasesSummary: CDK4/6抑制剂
- A3717 PF-5431 CitationTarget: Sphingosine kinases (SphKs)Summary: SphK1选择性抑制剂
- A8302 Tenovin-6Target: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT抑制剂,p53激活剂
- B1986 NedaplatinSummary: DNA合成抑制剂