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- B5963 7-Ethoxyresorufin中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮Target: Cytochrome P450 (CYP450)Summary: CYP1A特异性底物
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- A3967 Lapatinib Ditosylate中文名: 二苯磺酸拉帕替尼Target: EGFR|ErbB-2Summary: EGFR / HER2抑制剂
- B5864 Fruquintinib(HMPL-013)中文名: 呋喹替尼Target: VEGFRSummary: VEGFR1\2和3抑制剂
- A8253 PD 173074Target: VEGFR|FGFRSummary: FGFR抑制剂
- A8255 Sunitinib malate2 Citation中文名: 苹果酸舒尼替尼Target: VEGFRSummary: VEGFR/PDGFRβ/ KIT/ FLT3/RET/CSF-1R抑制剂
- B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
- A3870 TG 100801Target: VEGFR|FGFR|Src|Fyn kinaseSummary: 多激酶抑制剂
- B7590 Quinidine中文名: 奎尼丁Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)Summary: 降低Na+和K+通道电流
- A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2抑制剂