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- B3392 GSK269962ATarget: ROCK|RSK|MSKSummary: ROCK抑制剂
- A4228 Nutlin-3Target: MDM2Summary: MDM2 拮抗剂
- N1315 Parthenolide中文名: 小白菊内酯,欧苷菊Target: Histone Deacetylases (HDACs)|MDM2|DNA Methyltransferases|p53|5-HT
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A3762 RG71125 CitationTarget: MDM2Summary: MDM2抑制剂
- B7807 Netarsudil (AR-13324)Target: ROCKSummary: ROCK抑制剂
- B3523 Fasudil中文名: 法舒地尔Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 钙拮抗剂
- A5611 GSK429286ATarget: ROCKSummary: 选择性ROCK1/ROCK2抑制剂
- A3771 RKI-1447Target: ROCKSummary: ROCK1/ROCK2抑制剂
- A3825 SLx-21191 CitationTarget: ROCKSummary: ROCK2抑制剂