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- A4212 Pomalidomide (CC-4047)中文名: 泊马度胺Summary: 抗肿瘤/抗血管生成的免疫调制剂
- B2186 GSK2636771Target: PI3KSummary: PIK3抑制剂
- A3209 AXL1717中文名: 鬼臼毒素Target: Insulin-like growth factor receptors(IGFRs)Summary: IGF-1R抑制剂,口服有效。
- A8332 R788 disodium中文名: 福他替尼二钠盐Target: SykSummary: Syk的ATP竞争性抑制剂
- A1877 XAV-9391 CitationTarget: TNKSSummary: Tankyrase 1/2抑制剂
- A4317 Apremilast (CC-10004)中文名: 阿普斯特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂
- A8217 ICG 0011 CitationSummary: Wnt/β-catenin信号通路的抑制剂
- A5176 AS-605240Target: PI3KSummary: PI 3-Kγ选择性抑制剂
- A3721 PHA-767491Target: Cyclin-Dependent Kinases|MK2|Cdc7Summary: Cdc7 / CDK9抑制剂
- A4010 Salinosporamide A (NPI-0052, Marizomib)Target: ProteasomeSummary: 20S蛋白酶体抑制剂