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- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A4118 Hesperadin1 Citation中文名: 橙皮甙,橙皮苷Target: Aurora KinasesSummary: Aurora B抑制剂
- A3214 AZD11521 CitationTarget: Aurora KinasesSummary: Aurora B激酶抑制剂
- A4123 KW 2449Target: Aurora Kinases|FLT3|Bcr-AblSummary: 多重激酶抑制剂
- A3761 RG2833Target: HDACSummary: 脑渗透性HDAC抑制剂
- B5916 Chidamide1 CitationTarget: HDACSummary: HDAC抑制剂
- B2143 Tacrolimus (FK506)2 Citation中文名: 他克莫司Target: Peptidylprolyl isomerasesSummary: 大环内酯类钙调神经磷酸酶抑制剂,免疫抑制剂。
- A4489 TC-A 2317 hydrochlorideTarget: Aurora KinasesSummary: Aurora kinase A抑制剂
- A4116 Danusertib (PHA-739358)2 Citation中文名: 达鲁舍替Target: Aurora KinasesSummary: Aurora kinase(极光激酶)抑制剂