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- A1987 Ki164254 CitationTarget: LPA ReceptorsSummary: LPA受体拮抗剂
- B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
- A8253 PD 173074Target: VEGFR|FGFRSummary: FGFR抑制剂
- A3170 AM9662 CitationTarget: LPA ReceptorsSummary: LPA1拮抗剂
- B1591 Ki16198Target: LPA ReceptorsSummary: LPA拮抗剂
- A3969 Vatalanib1 Citation中文名: 瓦他拉尼碱Target: VEGFRSummary: 细胞渗透性VEGFR-1/-2抑制剂
- A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2抑制剂
- A3167 AM-095 free baseTarget: LPA ReceptorsSummary: 有效的LPA1受体拮抗剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂