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- A1905 3-Deazaneplanocin,DZNep6 Citation中文名: 3-去氮腺嘌呤ATarget: HydrolaseSummary: S-腺苷高半胱氨酸和EZH2抑制剂。
- A8626 ETP-46464Target: PI3K|mTOR|DNA-PK|ATM/ATRSummary: ATR抑制剂
- A4118 Hesperadin1 Citation中文名: 橙皮甙,橙皮苷Target: Aurora KinasesSummary: Aurora B抑制剂
- A4126 Aurora A Inhibitor I中文名: 极光A抑制剂ITarget: Aurora KinasesSummary: Aurora A抑制剂
- A4125 CYC116Target: Aurora Kinases|FLT3|VEGFRSummary: Aurora A/B抑制剂
- A4112 Barasertib (AZD1152-HQPA)3 Citation中文名: 巴拉塞替Target: Aurora KinasesSummary: Aurora Kinase B抑制剂
- A1769 KU-00606481 CitationTarget: PI3K|DNA-PKSummary: DNA-PK/PI3-K双重抑制剂
- B2178 BAY 80-6946 (Copanlisib)1 Citation中文名: 库潘尼西Target: PI3KSummary: PI3K抑制剂
- A3317 Clozapine N-oxide(CNO)1 Citation中文名: 氯氮平的N-氧化物Target: DREADD LigandsSummary: Clozapine代谢产物,用于化学遗传学
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂