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- A3347 Dabrafenib Mesylate (GSK-2118436)中文名: 达帕菲尼甲磺酸盐Target: RafSummary: BRAF(V600E)抑制剂
- A5071 GDC-08791 CitationTarget: RafSummary: B-Raf抑制剂
- A8226 TAK-632Target: RafSummary: Pan-RAF的强效选择性抑制剂
- A8616 A-674563Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSKSummary: Akt1 / PKA / CDK2的强效选择性抑制剂
- A3016 PLX-47201 CitationTarget: RafSummary: BRAF激酶抑制剂
- A8642 R5472 CitationTarget: Cyclin-Dependent KinasesSummary: CDK1/2/4抑制剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂
- A3004 Vemurafenib (PLX4032, RG7204)9 Citation中文名: 维罗非尼Target: RafSummary: BRAF激酶抑制剂
- A3197 AT7519 HydrochlorideTarget: Cyclin-Dependent KinasesSummary: CDK抑制剂
- A3009 Sorafenib2 Citation中文名: 索拉非尼Target: Raf|VEGFRSummary: Raf激酶和酪氨酸激酶抑制剂