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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A1302 GSK1904529ATarget: Insulin and Insulin-like ReceptorsSummary: IGF-1R/IR 选择性抑制剂
- A2614 Bortezomib (PS-341)24 Citation中文名: 硼替佐米Target: ProteasomeSummary: 蛋白酶体抑制剂
- A8513 Riluzole中文名: 力鲁唑Target: Voltage-gated Sodium (NaV) Channels|glutamate releaseSummary: 钠通道抑制剂
- A2578 Clasto-Lactacystin β-lactoneTarget: ProteasomeSummary: 蛋白酶体抑制剂
- B1492 PYR-412 CitationTarget: ProteasomeSummary: 泛素活化酶(E1)抑制剂
- A4011 ONX-0914 (PR-957)6 CitationTarget: ProteasomeSummary: 免疫蛋白酶体(immunoproteasome)抑制剂
- B1577 C6461 CitationTarget: p300Summary: HAT p300-CBP抑制剂
- A8163 AM 1142 CitationTarget: ProteasomeSummary: 20S蛋白酶体抑制剂