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- B6023 PD-1/PD-L1 inhibitor 2Target: PD-1/PD-L1 interactionSummary: PD-1/PD-L1相互作用的抑制剂
- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- A2678 SU112742 CitationTarget: METSummary: C-Met抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- A3573 LY2801653Target: METSummary: MET抑制剂
- A3368 DMAT2 CitationTarget: Pim|CK2|HIPK2|HIPK3Summary: CK2抑制剂
- A8325 Tivantinib (ARQ 197)2 CitationTarget: METSummary: C-Met抑制剂
- B2014 Probenecid1 Citation中文名: 丙磺舒Target: Organic anion transporters (OATs)|TRP ChannelSummary: 生物学活性