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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- A2678 SU112742 CitationTarget: METSummary: C-Met抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- A3573 LY2801653Target: METSummary: MET抑制剂
- A3302 CGI-17461 CitationTarget: BTKSummary: Btk抑制剂
- A3494 INCB3344Target: CCRSummary: CCR2趋化因子受体拮抗剂
- B6185 ACP-196中文名: 阿卡替尼Target: BTKSummary: 不可逆的BTK抑制剂
- A8325 Tivantinib (ARQ 197)2 CitationTarget: METSummary: C-Met抑制剂