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- B1533 BMS-3788061 CitationTarget: gp120/CD4Summary: Gp120/CD4抑制剂
- A4118 Hesperadin1 Citation中文名: 橙皮甙,橙皮苷Target: Aurora KinasesSummary: Aurora B抑制剂
- A4114 MLN8054Target: Aurora KinasesSummary: Aurora A激酶抑制剂
- A8315 NU7441 (KU-57788)4 CitationTarget: PI3K|DNA-PKSummary: DNA-PK抑制剂
- A4116 Danusertib (PHA-739358)2 Citation中文名: 达鲁舍替Target: Aurora KinasesSummary: Aurora kinase(极光激酶)抑制剂
- A8649 NU 7026Target: PI3K|DNA-PK|ATMSummary: 有效的、竞争性DNA-PK抑制剂
- B2172 PP121Target: mTOR|Eph Receptors|VEGFR|PDGFR|Bcr-Abl|Src|DNA-PK|P110|HckSummary: 酪氨酸激酶和磷酸肌醇激酶双重抑制剂
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂