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- N2791 Cucurbitacin E中文名: 葫芦素 ETarget: ActinSummary: 抑制肌动蛋白解聚
- A3012 Ruxolitinib (INCB018424)4 Citation中文名: 鲁索替尼Target: JAKSummary: JAK抑制剂
- A4069 BMS-707035Target: HIV IntegrasesSummary: HIV-1整合酶抑制剂
- A8204 Lopinavir中文名: 洛匹那韦Summary: HIV蛋白酶抑制剂
- B4492 HS-173Target: PI3KSummary: PI3Kα抑制剂
- B2307 LGK-9741 CitationSummary: PORCN抑制剂
- A2678 SU112742 CitationTarget: METSummary: C-Met抑制剂
- B1286 AZD7545Target: PDHKSummary: 有效的PDHK选择性抑制剂
- A4180 SRT1720 HCl3 CitationTarget: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT1激活剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂