FGFR
FGFRs (fibroblast growth factor receptors) are transmembrane tyrosine kinase receptor. It is involved in carcinogenesis and plays an important role in cell differentiation, survival and proliferation etc.
- B4985 CH5183284 (Debio-1347)Summary: 口服FGFR抑制剂
- A8706 BLU9931Target: FGFRSummary: 有效的FGFR4不可逆抑制剂
- B4904 ACTB-1003Target: VEGFR|FGFR|Tie-2|RSK|p70 S6KSummary: FGFR1抑制剂
- B7486 PD 161570Summary: FGFR抑制剂
- A8350 AZD4547Target: FGFRSummary: FGFR抑制剂
- A1367 AP26113Summary: 间变性淋巴瘤激酶(ALK)抑制剂
- A5467 Ponatinib (AP24534)1 CitationTarget: VEGFR|PDGFR|Bcr-Abl|FGFR|SrcSummary: pan-BCR-ABL抑制剂,多激酶抑制剂
- A2168 Dovitinib (TKI-258, CHIR-258)2 CitationTarget: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: 多靶点RTK抑制剂
- A8253 PD 173074Target: VEGFR|FGFRSummary: FGFR抑制剂
- A8252 Nintedanib (BIBF 1120)3 CitationTarget: VEGFR|PDGFR|FGFRSummary: VEGFR/PDGFR/FGFR抑制剂