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Signaling Pathways - Ribosomal s6 kinases (RSK) - Voltage-gated Sodium (NaV) Channels - c-Kit - Lactate Dehydrogenases (LDH)

27件产品中的 1-10

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  1. Isosafrole
    A8703 Isosafrole
    Target: Lactate Dehydrogenases (LDH)
    Summary: stiripentol类似物,有效的LDH抑制剂。
      ≥8.8 mg/mL
      insoluble in H2O
  2. Stiripentol
    A8704 Stiripentol
    中文名: 司替戊醇
    Target: Lactate Dehydrogenases (LDH)
    Summary: LDH抑制剂
      ≥9.9 mg/mL
      insoluble in H2O
  3. Dasatinib Monohydrate
    B5954 Dasatinib Monohydrate
    中文名: 达沙替尼一水合物
    Target: PDGFR|c-Kit|Bcr-Abl|Src
    Summary: ABL\SRC\KIT\PDGFR以及其它酪氨酸激酶抑制剂
      ≥25.3 mg/mL
      insoluble in H2O
  4. Dovitinib (TKI258) Lactate
    B5953 Dovitinib (TKI258) Lactate
    Target: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFR
    Summary: 酪氨酸激酶抑制剂(TKI)
      ≥10.62 mg/mL
      ≥168.2 mg/mL
  5. Pexidartinib (PLX3397)
    B5854 Pexidartinib (PLX3397)
     3 Citation
    中文名: 培西达替尼
    Target: FLT3|c-Kit|CSF1R
    Summary: CSF-1R抑制剂
      ≥20.9 mg/mL
      insoluble in H2O
  6. AZD2932
    B5835 AZD2932
    Target: FLT3|VEGFR|PDGFR|c-Kit
    Summary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
      Soluble in DMSO
  7. GSK 2837808A
    B4929 GSK 2837808A
    Target: Lactate Dehydrogenases (LDH)
    Summary: 乳酸脱氢酶A(LDHA)抑制剂
      ≥9.12 mg/mL
      insoluble in H2O
  8. ProTx II
    B5515 ProTx II
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: NaV1.7通道阻断剂
      Soluble to 1 mg/mL
  9. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  10. Amiloride HCl dihydrate
    B2268 Amiloride HCl dihydrate
    中文名: 盐酸阿米洛利二水合物
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Urokinases
    Summary: 有效上皮钠通道(ENaC)阻断剂
      ≥14.05 mg/mL
      insoluble in H2O

27件产品中的 1-10

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