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Signaling Pathways - Farnesoid X receptors (FXRs) - Pepsins - Hedgehog - Calpains

10 件产品

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  1. Obeticholic Acid
    B4888 Obeticholic Acid
     2 Citation
    中文名: 奥贝胆酸
    Target: Farnesoid X receptors (FXRs)
    Summary: FXR激动剂
      ≥21.5 mg/mL
      insoluble in H2O
  2. XL335
    B1528 XL335
    Target: Farnesoid X receptors (FXRs)
    Summary: FXR激动剂
      ≥20.4 mg/mL
      insoluble in H2O
  3. Lithocholic Acid
    A8463 Lithocholic Acid
    中文名: 石胆酸
    Target: Farnesoid X receptors (FXRs)|Vitamin D receptors (VDRs)|Pregnane X receptor(PXR)
    Summary: 维生素D受体PXR和FXR的激活剂
      ≥12.95 mg/mL
      insoluble in H2O
  4. PD 150606
    A4413 PD 150606
    Target: Calpains
    Summary: 非肽类钙蛋白酶抑制剂
      Soluble in DMSO
  5. MDL 28170
    A4412 MDL 28170
    Target: Cathepsins|Calpains
    Summary: Calpain和cathepsin B抑制剂
      ≥16.75 mg/mL
      insoluble in H2O
  6. Calpain Inhibitor I, ALLN
    A2602 Calpain Inhibitor I, ALLN
     2 Citation
    Target: Cathepsins|Calpains
    Summary: Calpain I/II/ B/L抑制剂
      ≥19.1 mg/mL
      insoluble in H2O
  7. E-64
    A2576 E-64
     2 Citation
    Target: Cathepsins|Calpains|Papains
    Summary: 半胱氨酸蛋白酶(cysteine protease)抑制剂
      ≥53.6 mg/mL
      ≥49.1 mg/mL
  8. GDC-0449 (Vismodegib)
    A3021 GDC-0449 (Vismodegib)
     1 Citation
    中文名: 维莫德吉
    Target: P-glycoprotein (P-gp)|Hedgehog
    Summary: Hedgehog拮抗剂
      ≥21.08 mg/mL
      insoluble in H2O
  9. Pepstatin A
    A2571 Pepstatin A
     1 Citation
    中文名: 抑肽素
    Target: Cathepsins|Renin|HIV proteases|Pepsins
    Summary: 天冬氨酸蛋白酶抑制剂
      ≥34.3 mg/mL
      insoluble in H2O
  10. Leupeptin, Microbial
    A2570 Leupeptin, Microbial
    中文名: 亮抑酶肽
    Target: Cathepsins|Calpains|Trypsins
    Summary: 丝氨酸和半胱氨酸蛋白酶抑制剂
      ≥24.7 mg/mL
      ≥54.4 mg/mL

10 件产品

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