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Signaling Pathways - endothelin receptor - Smoothened - angiogenesis - 5-HT Transporters

10 件产品

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  1. FR 139317
    B5082 FR 139317
    Target: endothelin receptor
    Summary: 选择性ETA内皮素受体拮抗剂
      Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
  2. Paroxetine HCl
    B2252 Paroxetine HCl
     1 Citation
    中文名: 盐酸帕罗西汀
    Target: 5-HT Transporters
    Summary: 抗抑郁药
      ≥36.73 mg/mL
      insoluble in H2O
  3. Desvenlafaxine
    B2236 Desvenlafaxine
    中文名: 去甲文拉法辛
    Target: 5-HT Transporters|Norepinephrine transporters
    Summary: 5-羟色胺(5-HT)和去甲肾上腺素(NE)再摄取抑制剂
      ≥13.2 mg/mL
  4. Amitriptyline HCl
    B2231 Amitriptyline HCl
    中文名: 盐酸阿米替林
    Target: Trk Receptors|5-HT2 Receptors|Norepinephrine transporter|5-HT Transporters
    Summary: 血清素/去甲肾上腺素受体/5-HT4/5-HT2抑制剂
      ≥15.69 mg/mL
      ≥43.9 mg/mL
  5. LDE225 (NVP-LDE225,Erismodegib)
    B2266 LDE225 (NVP-LDE225,Erismodegib)
     1 Citation
    中文名: 索尼德吉
    Target: Smoothened
    Summary: Smoothened抑制剂
      ≥24.3 mg/mL
      insoluble in H2O
  6. PF-04449913
    B3283 PF-04449913
    中文名: 格拉吉布
    Target: Smoothened
    Summary: Smoothened拮抗剂
      ≥20.15 mg/mL
      insoluble in H2O
  7. Cyclopamine
    A8340 Cyclopamine
     1 Citation
    中文名: 环巴胺
    Target: Smoothened
    Summary: Hedgehog (Hh)信号抑制剂
      ≥6.86 mg/mL
      insoluble in H2O
  8. LDE225 Diphosphate
    A3543 LDE225 Diphosphate
    Target: Smoothened
    Summary: Smo拮抗剂
      ≥27.85 mg/mL
      insoluble in H2O
  9. BMS-833923
    A3258 BMS-833923
    Target: Smoothened
    Summary: Smoothened抑制剂
      ≥47.4 mg/mL
      insoluble in H2O
  10. Lenalidomide (CC-5013)
    A4211 Lenalidomide (CC-5013)
    中文名: 来那度胺
    Target: angiogenesis
    Summary: 抗肿瘤药物,抑制血管生成。
      ≥100.8 mg/mL
      insoluble in H2O

10 件产品

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