Signaling Pathways - DREADD Ligands - Ubiquitin-activating Enzyme E1 - PDK-1 - MDM2
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- B1036 MLN49245 CitationTarget: NAE|Ubiquitin-activating Enzyme E1|SUMOylationSummary: NAE抑制剂
- B1244 PYZD-4409Target: Ubiquitin-activating Enzyme E1Summary: 泛素激活酶E1抑制剂
- A2846 OSU-03012 (AR-12)1 CitationTarget: PDK-1Summary: PDK1抑制剂
- A3762 RG71125 CitationTarget: MDM2Summary: MDM2抑制剂
- A3317 Clozapine N-oxide(CNO)1 Citation中文名: 氯氮平的N-氧化物Target: DREADD LigandsSummary: Clozapine代谢产物,用于化学遗传学
- A4228 Nutlin-3Target: MDM2Summary: MDM2 拮抗剂
- N1315 Parthenolide中文名: 小白菊内酯,欧苷菊Target: Histone Deacetylases (HDACs)|MDM2|DNA Methyltransferases|p53|5-HT