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Signaling Pathways - Calpains - Aldehyde Dehydrogenases - ROS1 - sodium channel

12件产品中的 1-10

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  1. Entrectinib
    B5859 Entrectinib
    中文名: 恩曲替尼
    Target: Trk Receptors|ALK|ROS1
    Summary: ALK激酶抑制剂
      ≥28.05 mg/mL
      insoluble in H2O
  2. PF-06463922
    B4882 PF-06463922
    中文名: 劳拉替尼
    Target: ALK|ROS1
    Summary: ALK/ROS1的强效选择性抑制剂
      ≥20.3 mg/mL
      insoluble in H2O
  3. Alda 1
    B5508 Alda 1
    Target: Aldehyde Dehydrogenases
    Summary: ALDH2激活剂
      ≥15.15 mg/mL
      insoluble in H2O
  4. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  5. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  6. PD 150606
    A4413 PD 150606
    Target: Calpains
    Summary: 非肽类钙蛋白酶抑制剂
      Soluble in DMSO
  7. MDL 28170
    A4412 MDL 28170
    Target: Cathepsins|Calpains
    Summary: Calpain和cathepsin B抑制剂
      ≥16.75 mg/mL
      insoluble in H2O
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. Disulfiram
    A4015 Disulfiram
    中文名: 双硫仑
    Target: Aldehyde Dehydrogenases
    Summary: 多巴胺β-羟化酶抑制剂
      ≥12 mg/mL
      insoluble in H2O
  10. Calpain Inhibitor I, ALLN
    A2602 Calpain Inhibitor I, ALLN
     2 Citation
    Target: Cathepsins|Calpains
    Summary: Calpain I/II/ B/L抑制剂
      ≥19.1 mg/mL
      insoluble in H2O

12件产品中的 1-10

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