Signaling Pathways - Renin - Protein Arginine Methyltransferases - iNOS - Glucagon Receptors - p53
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- B4989 EPZ015666Target: Protein Arginine MethyltransferasesSummary: PRMT5抑制剂
- B2215 Aliskiren Hemifumarate中文名: 阿利克仑半富马酸盐Target: ReninSummary: 肾素抑制剂
- A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: p53结合抑制剂,抗凋亡。
- A4483 PRIMA-1Target: p53Summary: BAX抑制剂
- A4481 PhiKan 083Target: p53Summary: P53稳定剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- A3220 Bardoxolone中文名: 巴多索隆Target: COX|iNOSSummary: 用于治疗慢性肾病,每天一次
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A4204 JNJ-26854165 (Serdemetan)1 CitationTarget: p53|HDM2 ubiquitin ligaseSummary: P53激活剂,阻断Mdm2-p53相互作用。
- A4206 Pifithrin-α (PFTα)2 CitationTarget: p53Summary: p53抑制剂