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Signaling Pathways - Selective - NUAK1 - Thymidine Phosphorylases - Cytochrome P450 (CYP450)

13件产品中的 1-10

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  1. WZ4003
    B1374 WZ4003
    Target: NUAK1|NUAK2
    Summary: NUAK1/2抑制剂
      ≥7.85 mg/mL
      insoluble in H2O
  2. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  3. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  4. Fluconazole
    B2094 Fluconazole
    中文名: 氟康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 三唑抗真菌剂
      ≥10.9 mg/mL
      insoluble in H2O
  5. Rifabutin
    B2126 Rifabutin
    中文名: 利福布丁
    Target: Cytochrome P450 (CYP450)
    Summary: 抗结核药物
      ≥42.35 mg/mL
      insoluble in H2O
  6. TOK-001
    A8623 TOK-001
    中文名: 加来特龙,伽来特隆
    Target: Androgen Receptors|Cytochrome P450 (CYP450)
    Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
      ≥12.4 mg/mL
      insoluble in H2O
  7. Thioridazine HCl
    A8537 Thioridazine HCl
    中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐
    Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 Receptors
    Summary: 钙通道蛋白抑制剂
      ≥20.35 mg/mL
      ≥6.78 mg/mL
  8. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  9. Tipiracil hydrochloride
    A3875 Tipiracil hydrochloride
    中文名: 盐酸替吡嘧啶
    Target: Thymidine Phosphorylases
    Summary: 胸苷磷酸化酶抑制剂
      insoluble in DMSO
      ≥13.25 mg/mL
  10. MRT67307 HCl
    A3635 MRT67307 HCl
    Target: TBK1|MARK1|NUAK1
    Summary: SIK/TBK-1/IKKe抑制剂
      ≥23.25 mg/mL
      ≥52.5 mg/mL

13件产品中的 1-10

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