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Signaling Pathways - ErbB-2 - RET - Adenosine Kinases - Cytochrome P450 (CYP450)

21件产品中的 11-20

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  1. Regorafenib
    A8236 Regorafenib
     4 Citation
    中文名: 瑞戈非尼
    Target: Raf|VEGFR|PDGFR|c-Kit|RET
    Summary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
      ≥25.04 mg/mL
      insoluble in H2O
  2. Lapatinib Ditosylate
    A3967 Lapatinib Ditosylate
    中文名: 二苯磺酸拉帕替尼
    Target: EGFR|ErbB-2
    Summary: EGFR / HER2抑制剂
      ≥24.3 mg/mL
      insoluble in H2O
  3. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  4. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  5. AST 487
    A3194 AST 487
     1 Citation
    Target: RET
    Summary: RET激酶抑制剂
      ≥26.5 mg/mL
      insoluble in H2O
  6. 5-Iodotubercidin
    A3125 5-Iodotubercidin
    中文名: 5-碘杀结核菌素
    Target: Adenosine Kinases
    Summary: 腺苷激酶抑制剂
      ≥83 mg/mL
      insoluble in H2O
  7. Clarithromycin
    A4322 Clarithromycin
    中文名: 克拉霉素
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A抑制剂
      ≥31.2 mg/mL
      insoluble in H2O
  8. Ketoconazole
    A4316 Ketoconazole
    中文名: 酮康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
      ≥23.4 mg/mL
      insoluble in H2O
  9. Cobicistat (GS-9350)
    A4313 Cobicistat (GS-9350)
    中文名: 可比司他
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A的选择性抑制剂
      ≥150.9 mg/mL
      insoluble in H2O
  10. Abiraterone acetate
    A8202 Abiraterone acetate
    中文名: 乙酸阿比特龙酯
    Target: Cytochrome P450 (CYP450)
    Summary: 细胞色素p450 17a1抑制剂
      ≥11.22 mg/mL
      insoluble in H2O

21件产品中的 11-20

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