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- A8319 Dacomitinib (PF299804, PF299)中文名: 达克替尼Target: ErbBSummary: HER抑制剂
- A3962 AZD1208Target: PimSummary: PIM激酶抑制剂
- A8375 AZD8931 (Sapitinib)中文名: 沙普替尼Target: EGFR|ErbBSummary: ErbB抑制剂
- A8218 Lapatinib2 Citation中文名: 拉帕替尼Target: ErbBSummary: EGFR/HER2抑制剂
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂
- B1543 Mubritinib (TAK 165)中文名: 木利替尼Target: ErbBSummary: HER2/ErbB2有效抑制剂
- B1255 AZ505Target: SMYD2Summary: SMYD2抑制剂
- A3368 DMAT2 CitationTarget: Pim|CK2|HIPK2|HIPK3Summary: CK2抑制剂
- A4193 SMI-4aTarget: PimSummary: Pim激酶抑制剂
- B2114 Mitoxantrone HCl中文名: 米托蒽醌Target: Pim|Topoisomerases|USP|HIV IntegrasesSummary: 拓扑异构酶II抑制剂