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- A4489 TC-A 2317 hydrochlorideTarget: Aurora KinasesSummary: Aurora kinase A抑制剂
- A4127 GSK1070916Target: Aurora KinasesSummary: Aurora B/C抑制剂
- A4115 JNJ-77066211 CitationTarget: Cyclin-Dependent Kinases|Aurora KinasesSummary: 有效的CDK/Aurora抑制剂
- A4335 Mildronate中文名: 米屈肼Target: Hydroxylases|carnitine reabsorptionSummary: GBB羟化酶抑制剂
- A8476 MK-2461Target: FLT3|PDGFR|MET|RonSummary: C-Met(野生型/突变型)抑制剂
- B2087 Ciclopirox中文名: 环吡酮胺Target: HydroxylasesSummary: 广谱抗真菌剂
- B4751 L-MimosineTarget: HydroxylasesSummary: 铁螯合剂和脯氨酰-4-羟化酶抑制剂
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A4116 Danusertib (PHA-739358)2 Citation中文名: 达鲁舍替Target: Aurora KinasesSummary: Aurora kinase(极光激酶)抑制剂