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- A4098 PCI-24781 (CRA-024781)Target: Histone Deacetylases (HDACs)Summary: Pan-HDAC抑制剂
- A8487 Nocodazole1 Citation中文名: 诺考达唑Target: Microtubules/TubulinsSummary: 微管蛋白产生抑制剂,抗肿瘤剂
- A1769 KU-00606481 CitationTarget: PI3K|DNA-PKSummary: DNA-PK/PI3-K双重抑制剂
- A3004 Vemurafenib (PLX4032, RG7204)9 Citation中文名: 维罗非尼Target: RafSummary: BRAF激酶抑制剂
- A5176 AS-605240Target: PI3KSummary: PI 3-Kγ选择性抑制剂
- N2791 Cucurbitacin E中文名: 葫芦素 ETarget: ActinSummary: 抑制肌动蛋白解聚
- N1359 Magnolol中文名: 厚朴酚Target: CB1 Receptors|NO Donors / Precursors|CB2 ReceptorsSummary: NO/TNF-α产生的抑制剂;抗真菌剂
- A8315 NU7441 (KU-57788)4 CitationTarget: PI3K|DNA-PKSummary: DNA-PK抑制剂
- A1748 Ramelteon1 Citation中文名: 雷美替胺Target: Melatonin ReceptorsSummary: MT1/MT2激动剂
- N2355 Madecassic acid中文名: 羟基积雪草酸