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- A4447 2,3-DCPE hydrochlorideTarget: Apoptosis InducersSummary: Bcl-XL蛋白表达下调剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A4302 Rosiglitazone maleate中文名: 马来酸罗格列酮Target: Insulin and Insulin-like ReceptorsSummary: PPARγ激动剂,有效的胰岛素敏化剂
- A8683 NVP-BHG712Target: Eph Receptors|VEGFRSummary: EphB4 抑制剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- B2172 PP121Target: mTOR|Eph Receptors|VEGFR|PDGFR|Bcr-Abl|Src|DNA-PK|P110|HckSummary: 酪氨酸激酶和磷酸肌醇激酶双重抑制剂
- B1519 Bazedoxifene HCl中文名: 盐酸巴多昔芬Target: Estrogen and Related ReceptorsSummary: 新的非甾体,基于吲哚的雌激素受体调节剂(SERM)
- B1506 Estradiol valerate中文名: 戊酸雌二醇Target: Estrogen and Related ReceptorsSummary: 雌激素受体激动剂
- B1515 Raloxifene HCl中文名: 盐酸雷洛昔芬Target: Estrogen and Related ReceptorsSummary: 雌激素受体(ER)调节剂