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- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: 有效的HER2选择性抑制剂
- B1106 VRT752271Target: ERKSummary: ERK1/ERK2 inhibitor
- A3965 BI 25361 CitationTarget: PLK|Bromodomain-containing proteins(BRDs)Summary: ATP竞争性的Plk1抑制剂
- A8616 A-674563Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSKSummary: Akt1 / PKA / CDK2的强效选择性抑制剂
- A3943 XMD8-92Target: ERKSummary: BMK1/ERK5抑制剂
- A3942 XMD17-109Target: ERKSummary: ERK-5抑制剂