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- A4447 2,3-DCPE hydrochlorideTarget: Apoptosis InducersSummary: Bcl-XL蛋白表达下调剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂
- A3009 Sorafenib2 Citation中文名: 索拉非尼Target: Raf|VEGFRSummary: Raf激酶和酪氨酸激酶抑制剂
- B6552 CGP 20712 dihydrochlorideTarget: adrenoceptorSummary: β1拮抗剂
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂
- A4121 SNS-314 MesylateTarget: Aurora KinasesSummary: Aurora A/B/C激酶抑制剂
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- B1407 Dabrafenib (GSK2118436)3 Citation中文名: 达拉菲尼Target: RafSummary: BRAF(V600)突变抑制剂
- A4122 PHA-680632Target: Aurora Kinases|PLK|FGFRSummary: Aurora激酶抑制剂