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- A3556 LKB1 (AAK1 dual inhibitor)Target: PimSummary: Pim-1激酶抑制剂
- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A3003 MDV3100 (Enzalutamide)12 Citation中文名: 恩杂鲁胺Target: Androgen ReceptorsSummary: 雄激素受体拮抗剂。
- A5065 Bicalutamide1 Citation中文名: 比卡鲁胺Target: Androgen ReceptorsSummary: 雄激素受体(Androgen receptor)拮抗剂
- A3149 AKT inhibitor VIII2 CitationTarget: AktSummary: 变构Akt激酶抑制剂
- A3440 Glyoxalase I inhibitorTarget: Glyoxalase ISummary: Glyoxalase I 抑制剂
- A4126 Aurora A Inhibitor I中文名: 极光A抑制剂ITarget: Aurora KinasesSummary: Aurora A抑制剂
- B3694 K-Ras(G12C) inhibitor 6Target: KRAS G12CSummary: K-Ras (G12C)抑制剂
- A4461 Bax inhibitor peptide V5Target: BaxSummary: Bax抑制剂