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- A8626 ETP-46464Target: PI3K|mTOR|DNA-PK|ATM/ATRSummary: ATR抑制剂
- A3724 PI-103 HydrochlorideTarget: PI3K|mTOR|DNA-PKSummary: DNA-PK / PI3-kinase / mTOR抑制剂
- A8610 6,2',4'-TrimethoxyflavoneTarget: Aryl hydrocarbon receptors (AHRs)Summary: 芳基烃受体拮抗剂
- B2178 BAY 80-6946 (Copanlisib)1 Citation中文名: 库潘尼西Target: PI3KSummary: PI3K抑制剂
- A2681 TGX-221Target: PI3KSummary: PI3K抑制剂
- A1905 3-Deazaneplanocin,DZNep6 Citation中文名: 3-去氮腺嘌呤ATarget: HydrolaseSummary: S-腺苷高半胱氨酸和EZH2抑制剂。
- B1288 RigosertibTarget: PI3K|PLKSummary: PI3K/PLK1抑制剂
- A3005 CAL-101 (Idelalisib, GS-1101)2 Citation中文名: 艾代拉里斯,艾代拉利司Target: PI3KSummary: PI3K抑制剂
- A3316 Clemizole hydrochloride中文名: 盐酸克立咪唑Target: Histamine H1 Receptors|TRPC channelSummary: H1组胺受体拮抗剂
- A1769 KU-00606481 CitationTarget: PI3K|DNA-PKSummary: DNA-PK/PI3-K双重抑制剂