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- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- B1810 Penfluridol中文名: 五氟利多Target: Voltage-gated Calcium Channels (CaV)Summary: 多巴胺受体拮抗剂
- A3604 Mibefradil中文名: 米贝拉地尔,米贝地尔,咪拉地尔,咪贝地尔Target: Voltage-gated Calcium Channels (CaV)Summary: 钙通道阻滞剂
- A2174 Lenvatinib (E7080)中文名: 乐伐替尼,仑伐替尼Target: VEGFR|PDGFR|RETSummary: VEGFR抑制剂
- B1505 Epiandrosterone中文名: 表雄酮Target: Voltage-gated Calcium Channels (CaV)Summary: 类固醇激素,具有弱雄激素活性
- B1988 Nifedipine2 Citation中文名: 硝苯地平Target: Voltage-gated Calcium Channels (CaV)Summary: L-型钙通道阻断剂
- B5854 Pexidartinib (PLX3397)3 Citation中文名: 培西达替尼Target: FLT3|c-Kit|CSF1RSummary: CSF-1R抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A3194 AST 4871 CitationTarget: RETSummary: RET激酶抑制剂
- B1572 LatrepirdineTarget: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptorSummary: 脑细胞死亡抑制剂