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- A8233 DMXAA (Vadimezan)2 Citation中文名: 2,5-己酮可可碱Target: DT-diaphorasesSummary: 肿瘤血管破坏剂,细胞凋亡诱导剂。
- B4888 Obeticholic Acid2 Citation中文名: 奥贝胆酸Target: Farnesoid X receptors (FXRs)Summary: FXR激动剂
- A4186 Bromosporine1 CitationTarget: BromodomainsSummary: Bromodomain抑制剂
- B1498 I-BET-7624 CitationTarget: BromodomainsSummary: BET抑制剂
- A1910 Bromodomain Inhibitor, (+)-JQ138 CitationTarget: BromodomainsSummary: BET bromodomain抑制剂。
- B1528 XL335Target: Farnesoid X receptors (FXRs)Summary: FXR激动剂
- B1531 (R)-baclofen中文名: (R)-巴氯芬Target: GABAB ReceptorsSummary: GABA受体激动剂
- B5086 CGP 55845 hydrochlorideTarget: GABAB ReceptorsSummary: GABAB受体拮抗剂
- B1012 MS436Target: BromodomainsSummary: BRD4抑制剂
- A4184 PFI-1 (PF-6405761)1 CitationTarget: BromodomainsSummary: BET抑制剂