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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- B6274 N-AcetyltryptamineTarget: Melatonin ReceptorsSummary: 褪黑激素受体调节剂
- A1748 Ramelteon1 Citation中文名: 雷美替胺Target: Melatonin ReceptorsSummary: MT1/MT2激动剂
- B2082 Camostat Mesilate中文名: 甲磺酸卡莫司他Target: Trypsin-like proteaseSummary: 胰蛋白酶样蛋白酶抑制剂
- B7407 Insulin (human) recombinant expressed in yeast中文名: 胰岛素Target: Insulin ReceptorsSummary: 内源性胰岛素受体激动剂
- B2014 Probenecid1 Citation中文名: 丙磺舒Target: Organic anion transporters (OATs)|TRP ChannelSummary: 生物学活性
- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: 有效的HER2选择性抑制剂